Ziritaxestat (Standard), CAS 1628260-79-6

Product Description: Ziritaxestat (Standard) is the analytical standard of Ziritaxestat. This product is intended for research and analytical applications. Ziritaxestat (GLPG1690) is a first-in-class autotaxin (ATX) inhibitor, with an IC50 of 131 nM and a Ki of 15 nM[1].

Formula: C30H33FN8O2S

References: [1]Desroy N, et al. Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis. J Med Chem. 2017 May 11;60(9):3580-3590.

CAS Number: 1628260-79-6

Molecular Weight: 588.70

Research Area: Inflammation/Immunology

Target: Phosphodiesterase (PDE);Reference Standards

• SKU: MEXHY-101772R-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-101772R-0
• Package Unit: Get quote
• Quantity Unit: STK