Product Description: FAK-IN-25 (4c) is a FAK inhibitor with an IC50 of 50.98 nM. FAK-IN-25 (4c) induces apoptosis and causes cell cycle arrest at G1 phase. FAK-IN-25 (4c) can be used in cancer research[1].
Formula: C22H13ClN4OS2
References: [1]Azza Ismail, et al. Exploring Thieno/Furo[2,3-b]pyridines as new scaffolds for potential FAK inhibition: Design, synthesis, biological evaluation and in silico studies. Bioorg Chem. 2025 Jun 1:159:108392.
Molecular Weight: 448.95
Research Area: Cancer
Target: Apoptosis;FAK