Linetastine, CAS 159776-68-8

Product Description: Linetastine is an orally active and potent 5-Lipoxygenase inhibitor. Linetastine shows antihistamine activity. Linetastine inhibits leukotriene production and antagonizes the effect of histamine. Linetastine inhibits the release of leukotrienes B4 and C4 from calcium ionophore-stimulated human leukocytes[1].

Applications: COVID-19-immunoregulation

Formula: C35H40N2O6

References: [1]Shizawa T, et al. 5-Lipoxygenase inhibitory and antihistamine activities of linetastine. Arzneimittelforschung. 1996 Nov;46(11):1072-6.

CAS Number: 159776-68-8

Molecular Weight: 584.70

Research Area: Inflammation/Immunology

Solubility: 10 mM in DMSO

Target: Histamine Receptor;Lipoxygenase

• SKU: MEXHY-123103-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-123103-5
• Package Unit: 5 mg
• Quantity Unit: STK