GSK973, CAS 2138473-38-6

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: (2S,3S)-2-(fluoromethyl)-2,3-dihydro-N7-methyl-N5-(1a,5ß,6ß)-3-oxabicyclo[3.1.0]hex-6-yl-3-phenyl-5,7-benzofurandicarboxamide

Purity: ≥98%

Formula Markup: C23H23FN2O4

Formula Weight: 410.438203

CAS Number: 2138473-38-6

Notes: A BET BD2 inhibitor (IC50s = 31.62, 15.85, 15.85, and 39.81 nM for BRD2, BRD3, BRD4, and BRDTBD2, respectively); selective for BD2 in BRD2, BRD3, BRD4, and BRDT over BD1 in the same BRDs (IC50s = >10,000 nM for all)

• SKU: CAY42057-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 42057-5
• Package Unit: 5 mg
• Quantity Unit: STK