MS049, CAS 1502816-23-0

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: N-methyl-4-(phenylmethoxy)-1-piperidineethanamine

Purity: ≥98%

Formula Markup: C15H24N2O

Formula Weight: 248.36394

CAS Number: 1502816-23-0

Notes: A selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM); less active against additional type I PRMTs (IC50s = >13, >22, and 1.6 µM for PRMT1, PRMT3, and PRMT8, respectively) and displays no inhibition against type II or type III PRMTs nor any additional methyltransferases or nonepigenetic targets tested; reduces H3R2me2a in HEK293 cells (IC50 = 0.97 µM) and also, unexpectedly, to reduce H4R3me2a in HEK293 cells

• SKU: CAY41105-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 41105-10
• Package Unit: 10 mg
• Quantity Unit: STK