Shelf life (days): 1460.0
Formulation: A solid
Formal Name: 2-nitro-N-[[trans-4-[[[(1,2,3,4-tetrahydro-2-naphthalenyl)methyl]amino]methyl]cyclohexyl]methyl]-benzenesulfonamide, monohydrochloride
Purity: ≥98%
Formula Markup: C25H33N3O4S / HCl
Formula Weight: 508.074
CAS Number: 191931-56-3
Notes: An antagonist of NPY receptor Y5 (Ki = 8 nM); selective for neuropeptide Y5 over Y1 receptors (Ki = >10,000 nM); suppresses colony formation by PC3 and DU145 cells at 10 and 20 µM; reduces tumor volume in a PC3 mouse xenograft model at 1, 3, and 10 mg/kg per day