Shelf life (days): 1460.0
Formulation: A solid
Formal Name: L-cysteinyl-L-threonyl-L-cysteinyl-L-asparaginyl-L-a-aspartyl-L-methionyl-L-threonyl-L-a-aspartyl-L-a-glutamyl-L-a-glutamyl-L-cysteinyl-L-leucyl-L-asparaginyl-L-phenylalanyl-L-cysteinyl-L-histidyl-L-glutaminyl-L-a-aspartyl-L-valyl-L-isoleucyl-L-tryptophan, cyclic (1?15),(3?11)-bis(disulfide), trifluoroacetate salt
Amino Acids: CTCNDMTDEECLNFCHQDVIW-OH
Purity: ≥98%
Formula Markup: C103H147N27O37S5 / XCF3COOH
Formula Weight: 2515.761
Notes: A peptide ETB receptor agonist; induces phosphatidyl inositol turnover in rat hippocampal slices (EC50 = ~10 nM); selectively binds to ETB over the ETA receptors (Kis = 0.023 and 4,200 nM for the rat hippocampal and atrial receptors, respectively); induces contractions in isolated dog saphenous vein segments and relaxation of isolated rabbit mesenteric artery segments; increases diastolic arterial pressure in pithed rats at 0.01-3 nmol/kg
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