Shelf life (days): 1460.0
Formulation: A solid
Formal Name: 2-bromo-N-[4-chloro-3-[[(3R)-1-methyl-3-pyrrolidinyl]oxy]phenyl]-4,5-dimethoxy-benzenesulfonamide
Purity: ≥95%
Formula Markup: C19H22BrClN2O5S
Formula Weight: 505.81116
CAS Number: 474960-44-6
Notes: A urotensin II receptor antagonist (Kis = 61, 17, 30, 65, and 56 nM for the human, monkey, cat, rat, and mouse receptors, respectively); reduces urotensin II-induced increases in the expression of IL1B, IL6, and VCAM1 in EA.hy926 cells at 1 µM; reduces urotensin II-induced adhesion of U937 monocytes to EA.hy926 cells at 1 µM