SGC2085, CAS 1821908-48-8

Product Description: SGC2085 is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1) with an IC50 of 50 nM. SGC2085 also selectively inhibits PRMT6 with an IC50 value of 5.2 μM, but not other PRMT proteins[1].

Applications: Cancer-programmed cell death

Formula: C19H24N2O2

References: [1]Ferreira de Freitas R, et al. Discovery of a Potent and Selective Coactivator Associated Arginine Methyltransferase 1 (CARM1) Inhibitor by Virtual Screening. J Med Chem. 2016 Jul 28;59(14):6838-47.

CAS Number: 1821908-48-8

Molecular Weight: 312.41

Compound Purity: 99.46

Research Area: Cancer

Solubility: DMSO : ≥ 32 mg/mL

Target: Histone Methyltransferase

• SKU: MEXHY-100565-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-100565-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK