SI-2 (hydrochloride), CAS 1992052-49-9

Product Description: SI-2 (EPH 116 hydrochloride) is a highly promising SRC-3 inhibitor (PPI), with IC50 values of 3-20 nM for breast cancer cell death. SI-2 (EPH 116 hydrochloride) has a much improved toxicity and pharmacokinetic profile, with acceptable oral availability[1].

Applications: Cancer-programmed cell death

Formula: C15H16ClN5

References: [1]Song X, et al. Development of potent small-molecule inhibitors to drug the undruggable steroid receptor coactivator-3. Proc Natl Acad Sci U S A. 2016 May 3;113(18):4970-5.

CAS Number: 1992052-49-9

Molecular Weight: 301.77

Compound Purity: 99.79

Research Area: Cancer

Solubility: DMSO : 5 mg/mL (ultrasonic)

Target: Estrogen Receptor/ERR;Others

• SKU: MEXHY-101447A-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-101447A-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK