Succinate/succinate receptor antagonist 1, CAS 2361972-29-2

Succinate/succinate receptor antagonist 1, CAS 2361972-29-2
SKU
MEXHY-150205-50
Packaging Unit
50 mg
Manufacturer
MedChemExpress

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Product Description: Succinate/succinate receptor antagonist 1 (compound 7a) is a succinate/succinate receptor antagonist. Succinate/succinate receptor antagonist 1 blocks succinate signaling in gingival tissue. Succinate/succinate receptor antagonist 1 inhibits the activation of succinate receptor 1 (SucnRl) with an IC50 value of 20 μΜ. Succinate/succinate receptor antagonist 1 can be used for the research of periodontal disease[1].

Applications: COVID-19-immunoregulation

Formula: C17H15N3O

References: [1]LI, Xin, et al. PERIODONTAL DISEASE THERAPY. WO2019136022. 2020.

CAS Number: 2361972-29-2

Molecular Weight: 277.32

Compound Purity: 99.46

Research Area: Inflammation/Immunology

Solubility: DMSO : 25 mg/mL (ultrasonic)

Target: Succinate Receptor 1
More Information
SKU MEXHY-150205-50
Manufacturer MedChemExpress
Manufacturer SKU HY-150205-50
Package Unit 50 mg
Quantity Unit STK
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