Product Description: Usmarapride (SUVN-D4010) free base is a potent, selective, orally active and brain penetrant 5-HT4 receptor partial agonist (EC50=44 nM). Usmarapride (SUVN-D4010) free base can be used for the research of cognitive deficits associated with Alzheimer's disease[1].
Applications: Neuroscience-Neurodegeneration
Formula: C21H29N5O2
References: [1]Nirogi R, et al. Discovery and Preclinical Characterization of Usmarapride (SUVN-D4010): A Potent, Selective 5-HT4 Receptor Partial Agonist for the Treatment of Cognitive Deficits Associated with Alzheimer's Disease. J Med Chem. 2021;64(15):10641-10665.
CAS Number: 1428862-32-1
Molecular Weight: 383.49
Compound Purity: 99.91
Research Area: Neurological Disease
Solubility: DMSO : ≥ 100 mg/mL
Target: 5-HT Receptor