Vasopressin V2 receptor antagonist 2

Product Description: Vasopressin V2 receptor antagonist 2 (Compound 33) is an antagonist of the arginine vasopressin V2 receptor (V2R) with a Ki value of 6.2 nM. Vasopressin V2 receptor antagonist 2 can effectively reduce cAMP levels, thereby inhibiting the growth of renal cysts[1].

Applications: Metabolism-protein/nucleotide metabolism

Formula: C62H91FN16O11

References: [1]Xiong X, et al. Long-Residence Time Peptide Antagonist for the Vasopressin V₂ Receptor to Treat Autosomal Dominant Polycystic Kidney Disease. J Med Chem. 2024;67(7):5935-5944.

Molecular Weight: 1255.48

Compound Purity: 99.81

Research Area: Metabolic Disease

Solubility: DMSO : 12.5 mg/mL (ultrasonic;warming;heat to 60°C)

Target: Vasopressin Receptor

• SKU: MEXHY-162394-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-162394-5
• Package Unit: 5 mg
• Quantity Unit: STK