Product Description: Velnacrine (HP 029 free base) is an inhibitor for acetylcholinesterase (AChE), with an IC50 of 3.27 μM. Velnacrine reverses the Scopolamine (HY-N0296)-induced amnesia in rat models, and exhibits acute toxicity with LD50 of 65 mg/kg[1].
Applications: Neuroscience-Neuromodulation
Formula: C13H14N2O
References: [1]Tabarrini O, et al., Velnacrine thiaanalogues as potential agents for treating Alzheimer's disease. Bioorg Med Chem. 2001 Nov;9(11):2921-8.
CAS Number: 124027-47-0
Molecular Weight: 214.26
Research Area: Neurological Disease
Target: Cholinesterase (ChE)