Product Description: Vipadenant (BIIB-014; CEB-4520) is an adenosine receptor antagonist, with Kis of 1.3 nM and 68 nM for A2A and A1, respectively.
Applications: Neuroscience-Neuromodulation
Formula: C16H15N7O
References: [1]Jones N, et al. A2A receptor antagonists do not induce dyskinesias in drug-naive or L-dopa sensitized rats. Brain Res Bull. 2013 Sep;98:163-9./[2]Brian C. Shook, et al. Adenosine A2A Receptor Antagonists and Parkinson’s Disease. ACS Chem Neurosci. 2011 Oct 19; 2(10): 555-567.
CAS Number: 442908-10-3
Molecular Weight: 321.34
Compound Purity: 98.02
Research Area: Neurological Disease
Solubility: DMSO : 31 mg/mL (ultrasonic;warming)
Target: Adenosine Receptor