Y06036, CAS 1832671-96-1

Product Description: Y06036 is a potent and selective BET inhibitor, which binds to the BRD4(1) bromodomain with Kd value of 82 nM[1]. Antitumor activity[1].

Applications: Neuroscience-Neuromodulation

Formula: C16H15BrN2O5S

References: [1]Zhang M, et al. Structure-Based Discovery and Optimization of Benzo[ d]isoxazole Derivatives as Potent and Selective BET Inhibitors for Potential Treatment of Castration-Resistant Prostate Cancer (CRPC). J Med Chem. 2018 Apr 12;61(7):3037-3058.

CAS Number: 1832671-96-1

Molecular Weight: 427.27

Compound Purity: 98.57

Research Area: Cancer

Solubility: DMSO : 130 mg/mL (ultrasonic)

Target: Epigenetic Reader Domain

• SKU: MEXHY-111502-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-111502-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK