ZEN-2759, CAS 1616400-50-0

Product Description: ZEN-2759 is a potent BET (Bromodomain and Extra-Terminal Domain) inhibitor, with IC50 values of 0.23, 0.08 and 0.28 μM for BRD4(BD1), BRD4(BD2), and BRD4(BD1BD2), respectively[1].

Applications: Cancer-programmed cell death

Formula: C17H16N2O2

References: [1]Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.

CAS Number: 1616400-50-0

Molecular Weight: 280.32

Compound Purity: 99.51

Research Area: Cancer

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Epigenetic Reader Domain

• SKU: MEXHY-129201-100
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-129201-100
• Package Unit: 100 mg
• Quantity Unit: STK